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PI3K/AKT-IN-1

Product Specifications

CAS Number

3033069-84-7

Target

PI3K

Applications

PI3K/Akt/mTOR

Molecular Formula

C23H23N5O4S

Additionnal Information

PI3K/AKT-IN-1 is a dual-acting inhibitor of PI3K/AKT pathway with an IC50 of 6.99 μM, 4.01 μM, and 3.36 μM, for PI3Kδ, PI3Kγ and AKT-1 respectively. It also induces S-phase cell cycle arrest, caspase-3-dependent apoptosis, exhibiting strong potential against breast cancer and leukemia.

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