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PFI-6

Product Specifications

CAS Number

2675452-91-0

Target

Others

Applications

Others

Molecular Formula

C22H21N3O4

Additionnal Information

PFI-6 is a selective MLLT1/3 probe that targets the YEATS domain of MLLT1 (ENL/YEATS1) and MLLT3 (AF9/YEATS3) with IC50 values of 140 nM and 160 nM for MLLT1 and MLLT3, respectively. PFI-6 demonstrates increased affinity and selectivity for MLLT1/3 than other human YEATS domain proteins (YEATS2/4) .

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