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Aticaprant

Product Specifications

CAS Number

1174130-61-0

Synonyms

CERC-501, LY-2456302

Target

Opioid Receptor

Applications

Neuronal Signaling

Molecular Formula

C26H27FN2O2

Additionnal Information

Aticaprant (CERC-501, LY-2456302) is a potent, orally bioavailable, centrally-penetrant antagonist of the kappa opioid receptor with a Ki of 0.807 nM. It exhibits an antidepressant effect with the potential to treat major depressive disorder (MDD) .

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