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BIIB129

Product Specifications

CAS Number

2770960-52-4

Target

BTK

Applications

Protein Tyrosine Kinase

Molecular Formula

C19H22N6O2

Additionnal Information

BIIB129, is a unique brain-penetrant covalent inhibitor of Bruton’s tyrosine kinase (BTK), with high kinome selectivity. It exhibits efficacy in targeting B-cell proliferation in the central nervous system (CNS), making it a promising immunomodulatory therapy for multiple sclerosis (MS) .

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