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FIDAS-5

Product Specifications

CAS Number

1391934-98-7

Target

Transferase

Applications

Metabolism

Molecular Formula

C15H13ClFN

Additionnal Information

FIDAS-5 is a potent and orally active inhibitor of methionine S-adenosyltransferase 2A (MAT2A) with an IC50 value of 2.1 μM, respectively. FIDAS-5 effectively competes against S-adenosylmethionine (SAM) for MAT2A binding. FIDAS-5 also demonstrates anticancer activity.

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