FIDAS-5
Product Specifications
CAS Number
1391934-98-7
Target
Transferase
Applications
Metabolism
Molecular Formula
C15H13ClFN
Additionnal Information
FIDAS-5 is a potent and orally active inhibitor of methionine S-adenosyltransferase 2A (MAT2A) with an IC50 value of 2.1 μM, respectively. FIDAS-5 effectively competes against S-adenosylmethionine (SAM) for MAT2A binding. FIDAS-5 also demonstrates anticancer activity.
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