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RP-102124

Product Specifications

CAS Number

2924486-45-1

Target

Rho

Applications

Cell Cycle

Molecular Formula

C23H16ClN5O2

Additionnal Information

RP-102124 is a first-in-class allosteric inhibitor of multi-Rac with activity against oncogenic Rac1b. RP-102124 is orally bioavailable and exhibits dose-dependent inhibition of tumor growth in xenograft models. It exhibits potent inhibition of phenotypic characteristics of Rac signaling such as cell migration and cytoskeletal rearrangements.

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