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L-778123 hydrochloride

Product Specifications

CAS Number

253863-00-2

Target

Telomerase

Applications

DNA Damage/DNA Repair

Molecular Formula

C22H20ClN5O.ClH

Additionnal Information

L-778123 hydrochloride is a potent dual inhibitor of farnesyl protein transferase (FPTase) with an IC50 of 2 nM and geranylgeranyl protein transferase I (GGPTase-I) with an IC50 of 98 nM. It also displays promising anti-leukemia activity.

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