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GLPG0187

Product Specifications

CAS Number

1320346-97-1

Target

Integrin

Applications

Cytoskeletal Signaling

Molecular Formula

C29H37N7O5S

Additionnal Information

GLPG0187 is a broad-spectrum antagonist of integrin receptor. It inhibits αvβ1-integrin with an IC50 value of 1.3 nM. GLPG0187 also inhibits migrasome biogenesis without cytotoxicity. GLPG0187 exhibits potent antitumor activity.

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