BGB-3245 (Brimarafenib)
Product Specifications
CAS Number
1643326-82-2
Synonyms
Brimarafenib, Brimarafenibum
Target
Raf
Applications
MAPK
Molecular Formula
C24H17F3N4O4
Additionnal Information
BGB-3245 (Brimarafenib, Brimarafenibum) is an inhibitor of Raf kinase. BGB-3245 displays potent effects against different RAF isoforms, including BRAF Class I/II/III mutations, BRAF fusions, and heterodimerization with CRAF in preclinical models. It also exhibits antineoplastic effects.
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