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AG 825

Product Specifications

CAS Number

149092-50-2

Synonyms

Tyrphostin AG-825

Target

EGFR

Applications

Protein Tyrosine Kinase

Molecular Formula

C19H15N3O3S2

Additionnal Information

AG-825 (Tyrphostin AG-825) is a potent and selective inhibitor of ErbB2 with IC50 values of 0.15 μM. It also inhibits PDGFR autophosphorylation with IC50 value of 40 μM. It exhibits anti-cancer activity and significantly induces apoptosis in cancer cells.

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