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AG 1295

Product Specifications

CAS Number

71897-07-9

Target

PDGFR

Applications

Protein Tyrosine Kinase

Molecular Formula

C16H14N2

Additionnal Information

AG 1295 is a selective and specific inhibitor of platelet-derived growth factor receptor (PDGFR) tyrosine-kinase. It inhibits PDGFR autophosphorylation with IC50 values of 0.3-0.5 μM in membrane autophosphorylation assays, respectively.

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