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GLPG3970

Product Specifications

CAS Number

2403733-82-2

Target

SIK

Applications

Immunology & Inflammation

Molecular Formula

C25H27F3N4O4

Additionnal Information

GLPG3970 (compound 32) is a dual inhibitor of SIK2 and SIK3, with IC50 of 282.8 nM, 7.8 nM and 3.8 nM for SIK1, SIK2 and SIK3, respectively. It has the potential to treat autoimmune and inflammatory diseases.
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