What is the catalog number for Tunlametinib?

The catalog number for Tunlametinib is E1943-1g.

What sizes are available for Tunlametinib?

Tunlametinib is available in the following size(s): 1 g.

Is Tunlametinib in stock?

Tunlametinib is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Tunlametinib?

Tunlametinib is manufactured by Bimake.

What is the estimated delivery time for Tunlametinib?

Estimated delivery time for Tunlametinib is approximately 15 business day(s), depending on your location.

Tunlametinib

Product Specifications

CAS Number

1801756-06-8

Synonyms

HL-085

Target

MEK

Applications

Protein Tyrosine Kinase

Molecular Formula

C16H12F2IN3O3S

Additionnal Information

Tunlametinib (HL-085) is a highly selective and oral inhibitor of MEK1/2 with an IC50 of 1.9 nM for MEK1, with the potential to treat RAS/RAF mutant cancers. It also induces cell cycle arrest at the G0/G1 phase and promotes apoptosis in a dose-dependent manner. It also exhibits antitumor activity in patients with advanced NRAS-mutant melanoma.