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BGB-8035

Product Specifications

CAS Number

2283349-24-4

Target

BTK

Applications

Protein Tyrosine Kinase

Molecular Formula

C24H31N5O4

Additionnal Information

BGB-8035 is an orally active, highly selective inhibitor of Bruton's tyrosine kinase (BTK) with IC50 values of 1.1 nM for BTK, respectively. BGB-8035 exhibits antitumor and anti-arthritis activity and displays potential for its use in research of B-cell malignancies and autoimmune diseases.
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