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Zongertinib

Product Specifications

CAS Number

2728667-27-2

Synonyms

BI 1810631, BI 764532

Target

HER2

Applications

Protein Tyrosine Kinase

Molecular Formula

C29H29N9O2

Additionnal Information

Zongertinib (BI 1810631, BI 764532) is a selective and potent inhibitor of human HER2 and EGFR tyrosine kinase that covalently binds to both wild-type and mutated HER2 receptors, including exon 20 insertion mutations, while sparing EGFR signaling. It exhibits effective and tolerable oral treatment for patients with HER2 aberration-positive solid tumors.

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