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BRD7389

Product Specifications

CAS Number

376382-11-5

Target

S6 Kinase

Applications

MAPK

Molecular Formula

C24H18N2O2

Additionnal Information

BRD7389 is an inhibitor of RSK family kinases with IC50 of 1.5 μM, 2.4 μM, and 1.2 μM for RSK1, RSK2, and RSK3, respectively. BRD7389 also increases β-cell–specific gene expression in primary human islet cells.

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