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LY2780301

Product Specifications

CAS Number

1226801-23-5

Target

Akt

Applications

PI3K/Akt/mTOR

Molecular Formula

C25H27F4N7O

Additionnal Information

LY2780301 is a highly selective adenosine triphosphate (ATP) -competitive dual inhibitor of p70S6K and Akt. LY2780301 binds to Akt, inhibiting its activity, which consequently blocks the PI3K/Akt signaling pathway which leads to reduced cell proliferation and the initiation of apoptosis in tumor cells.

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