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MKI-1

Product Specifications

CAS Number

1190277-80-5

Synonyms

MASTL Kinase Inhibitor-1

Target

Serine/threonin kinase

Applications

Cell Cycle

Molecular Formula

C18H14N4O

Additionnal Information

MKI-1 (MASTL Kinase Inhibitor-1) is an small-molecule inhibitor of MASTL (microtubule-associated serine/threonine kinase-like) with an IC50 9.9 μM in kinase assay. It also exerts antitumor and radiosensitizer activities through PP2A-mediated c-Myc inhibition in breast cancer models.

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