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TC-S 7009

Product Specifications

CAS Number

1422955-31-4

Target

HIF

Applications

Angiogenesis

Molecular Formula

C12H6ClFN4O3

Additionnal Information

TC-S 7009 is a potent and selective inhibitor of HIF-2α with a Kd value of 81 nM. TC-S 7009 is more selective for HIF-2α than HIF-1α. It disrupts HIF-2α heterodimerization, decreases DNA-binding activity, and reduces HIF-2α target gene expression.

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