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VT103

Product Specifications

CAS Number

2290608-13-6

Target

TEAD

Applications

Hippo

Molecular Formula

C18H17F3N4O2S

Additionnal Information

VT103 is an orally active and selective inhibitor of TEAD1 protein palmitoylation with anti-proliferative and anti-tumor activity. It also inhibits YAP/TAZ-TEAD promoted gene transcription, blocks TEAD auto-palmitoylation and disrupts interaction between YAP/TAZ and TEAD.

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