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Bezuclastinib

Product Specifications

CAS Number

1616385-51-3

Synonyms

CGT9486, PLX 9486

Target

C-Kit

Applications

Protein Tyrosine Kinase

Molecular Formula

C19H17N5O

Additionnal Information

Bezuclastinib (CGT9486; PLX 9486) is a potent inhibitor of c-kit and c-kit D816V with an IC50 value of <1 μM. Bezuclastinib is also an inhibitor of tyrosine kinase.

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