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BI-0474

Product Specifications

CAS Number

2750570-55-7

Target

Ras

Applications

Apoptosis

Molecular Formula

C30H37N9O2S

Additionnal Information

BI-0474 is a potent inhibitor of KRASG12C with an IC50 value of 7.0 nM. It inhibits GDP-KRAS::SOS1 protein-protein interactions. It exhibits anti-proliferative and anti-tumour activity and can be used in cancer research.

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