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Glesatinib

Product Specifications

CAS Number

936694-12-1

Synonyms

MGCD265

Target

C-Met

Applications

Protein Tyrosine Kinase

Molecular Formula

C31H27F2N5O3S2

Additionnal Information

Glesatinib (MGCD265) is an orally bioavailable potent dual inhibitor of c-MET and SMO. Glesatinib counteracts P-glycoprotein (P-gp) mediated multidrug resistance (MDR) in non-small cell lung cancer (NSCLC) .

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