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Ziftomenib

Product Specifications

CAS Number

2134675-36-6

Synonyms

KO-539

Target

MLL

Applications

Epigenetics

Molecular Formula

C33H42F3N9O2S2

Additionnal Information

Ziftomenib (KO-539) is an oral inhibitor of menin targeting the menin–KMT2A protein-protein interaction. It exhibits antileukemic activity and induces apoptosis of acute myeloid leukemia (AML) cells.

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