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VIT-2763

Product Specifications

CAS Number

2095668-10-1

Target

Others

Applications

Others

Molecular Formula

C21H21FN6O2

Additionnal Information

VIT-2763 is an oral small-molecule inhibitor of ferroportin. It displaces TMR-hepcidin from ferroportin with an IC50 of 24 nM. It also ameliorates anemia, enhances erythropoiesis, and reduces organ iron loading in the Hbbth3/+ β-thalassemia intermedia disease model.

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