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EZM0414

Product Specifications

CAS Number

2411748-50-8

Target

SETD

Applications

Epigenetics

Smiles

CC (=O) N1CCN (CC1) C2CCCC (C2) NC (=O) C3=CC4=C (F) C=CC (=C4[NH]3) C

Molecular Formula

C22H29FN4O2

Additionnal Information

EZM0414 is a potent, selective, and orally bioavailable inhibitor of Histone-lysine N-methyltransferase SETD2.

Storage Conditions

3 years -20°C powder

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