What is the catalog number for GSK215?

The catalog number for GSK215 is E1113-5mg.

What sizes are available for GSK215?

GSK215 is available in the following size(s): 5 mg.

GSK215 is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures GSK215?

GSK215 is manufactured by Bimake.

What is the estimated delivery time for GSK215?

Estimated delivery time for GSK215 is approximately 15 business day(s), depending on your location.

GSK215

Product Specifications

CAS Number

2743427-26-9

Target

FAK

Applications

Protein Tyrosine Kinase

Smiles

CNC (=O) C1=C (NC2=CC (=NC=C2C (F) (F) F) NC3=C (OC) C=C (C=C3) N4CCN (CC4) CC (=O) NC (C (=O) N5CC (O) CC5C (=O) NC (C) C6=CC=C (C=C6) C7=C (C) N=CS7) C (C) (C) C) C=CC=C1

Molecular Formula

C50H59F3N10O6S

Additionnal Information

GSK215 is a potent and selective PROTAC focal adhesion kinase (FAK) degrader, which exerts FAK degradation in A549 non-small-cell lung cancer cells with DC50 of 1.3 nM by a strong time-dependence way and maximal degradation (Dmax) near the limit of the assay quantification (Dmax 99%) .