What is the catalog number for Relacorilant (CORT125134)?

The catalog number for Relacorilant (CORT125134) is E1091-10mM/1mL.

What sizes are available for Relacorilant (CORT125134)?

Relacorilant (CORT125134) is available in the following size(s): 10 mM/1mL.

Is Relacorilant (CORT125134) in stock?

Relacorilant (CORT125134) is currently made to order / not held in immediate stock. Contact us for lead time.

Who manufactures Relacorilant (CORT125134)?

Relacorilant (CORT125134) is manufactured by Bimake.

What is the estimated delivery time for Relacorilant (CORT125134)?

Estimated delivery time for Relacorilant (CORT125134) is approximately 15 business day(s), depending on your location.

Relacorilant (CORT125134)

Product Specifications

CAS Number

1496510-51-0

Target

Glucocorticoid Receptor

Applications

Endocrinology & Hormones

Smiles

C[N]1C=C (C=N1) [S; v6] (=O) (=O) N2CCC3=CC4=C (CC3 (C2) C (=O) C5=CC (=CC=N5) C (F) (F) F) C=N[N]4C6=CC=C (F) C=C6

Molecular Formula

C27H22F4N6O3S

Additionnal Information

Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.