Relacorilant (CORT125134)
Product Specifications
CAS Number
1496510-51-0
Target
Glucocorticoid Receptor
Applications
Endocrinology & Hormones
Smiles
C[N]1C=C (C=N1) [S; v6] (=O) (=O) N2CCC3=CC4=C (CC3 (C2) C (=O) C5=CC (=CC=N5) C (F) (F) F) C=N[N]4C6=CC=C (F) C=C6
Molecular Formula
C27H22F4N6O3S
Additionnal Information
Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
Storage Conditions
3 years -20°C powder
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