Lartesertib (M4076)
Product Specifications
CAS Number
2495096-26-7
Target
ATM/ATR
Applications
PI3K/Akt/mTOR
Molecular Formula
C23H21FN6O3
Additionnal Information
Lartesertib (M4076) inhibits Ataxia telangiectasia-mutated (ATM) kinase activity with a sub-nanomolar potency and shows remarkable selectivity against other protein kinases, suppresses DSB repair, clonogenic cancer cell growth, and potentiates antitumor activity of ionizing radiation in cancer cell lines.
Storage Conditions
3 years -20°C powder
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