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SY-5609

Product Specifications

CAS Number

2417302-07-7

Synonyms

CDK7-IN-3

Target

CDK

Applications

Cell Cycle

Molecular Formula

C23H26F3N6OP

Additionnal Information

SY-5609 (CDK7-IN-3) is an orally active and highly selective inhibitor of CDK7 with a KD value of 0.065 nM. SY-5609 exhibits poor inhibition on CDK2, CDK9, CDK12. SY-5609 displays antitumor activity and can induce apoptosis in tumor cells.
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