Zapnometinib (PD0184264)
Product Specifications
CAS Number
303175-44-2
Synonyms
ATR-002
Target
MEK
Applications
Protein Tyrosine Kinase
Smiles
OC (=O) C1=C (NC2=C (Cl) C=C (I) C=C2) C (=C (F) C=C1) F
Molecular Formula
C13H7ClF2INO2
Additionnal Information
Zapnometinib (PD0184264, ATR-002), an major active metabolite of CI-1040, is a novel MEK inhibitor with an IC50 of 5.7 nM.
Storage Conditions
3 years -20°C powder
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