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PF-9363

Product Specifications

CAS Number

2569009-58-9

Synonyms

CTx-648

Target

Histone Acetyltransferase

Applications

Epigenetics

Smiles

COC1=CC (=CC2=C1C (=NO2) N[S] (=O) (=O) C3=C (OC) C=CC=C3OC) C[N]4C=CC=N4

Molecular Formula

C20H20N4O6S

Additionnal Information

PF-9363 is a potent and selective KAT6A/6B inhibitor with Ki of 0.41 nM and 1.2 nM for KAT6A and KAT6B, respectively. PF-9363 displays potent anti-tumor activity in ER+ breast cancer models.

Storage Conditions

3 years -20°C powder

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