CRTh2 antagonist 2
CRTh2 antagonist 2 is selective and potent CRTH2 antagonist extracted from patent US20140148470A1, compound Example 1, has an IC50 of ≤10 nM. CRTh2 antagonist 2 can be used in research of androgenic alopecia[1].
Product Specifications
CAS Number
780763-95-3
UNSPSC
12352005
Target
Prostaglandin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology
Assay Protocol
https://www.medchemexpress.com/crth2-antagonist-2.html
Purity
99.78
Solubility
DMSO : 125 mg/mL (ultrasonic)
Smiles
O=C(O)CC1=C(N(C)C)N=C(CC2=CC=C(NC(C3=CC=C4C=CC=CC4=C3)=O)C=C2)N=C1Cl
Molecular Formula
C26H23ClN4O3
Molecular Weight
474.94
References & Citations
[1]Andreas Schnapp, et al. Pyrimidine compounds for treating hairloss. US20140148470A1.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
DP
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