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PF-06273340

Product Specifications

CAS Number

1402438-74-7

SKU

C18177-25mg

Target

Trk receptor

Applications

Protein Tyrosine Kinase

Smiles

CC (C) (CO) N1C=C (C2=CN=C (N=C21) N) C (=O) C3=CC (=CN=C3) NC (=O) CC4=NC=C (C=C4) Cl

Molecular Formula

C23H22ClN7O3

Additionnal Information

PF-06273340 is a highly potent, kinases elective, well-tolerated pan-Trk inhibitor with IC50 values of 6, 4, 3 nM for TrkA, TrkB, Trk C, respectively.

Storage Conditions

2 years -80 in solvent

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