What is the catalog number for Birabresib (OTX015)?

The catalog number for Birabresib (OTX015) is C17931.

What sizes are available for Birabresib (OTX015)?

Birabresib (OTX015) is available in the following size(s): 100 mg.

Is Birabresib (OTX015) in stock?

Birabresib (OTX015) is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for Birabresib (OTX015)?

Birabresib (OTX015) is requires dry ice shipping.

Birabresib (OTX015)

Product Specifications

CAS Number

202590-98-5

Synonyms

MK 8628

SKU

C17931-100mg

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CC1=C (SC2=C1C (=NC (C3=NN=C (N32) C) CC (=O) NC4=CC=C (C=C4) O) C5=CC=C (C=C5) Cl) C

Molecular Formula

C25H22ClN5O2S

Additionnal Information

Birabresib (OTX015, MK 8628) is a potent BET bromodomain inhibitor with EC50 ranging from 10 to 19 nM for BRD2, BRD3, and BRD4 in cell-free assays. Birabresib inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.