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AGI-6780

Product Specifications

CAS Number

1432660-47-3

SKU

C17911-5mg

Target

Dehydrogenase

Applications

Metabolism

Smiles

C1CC1NS (=O) (=O) C2=CC (=C (C=C2) C3=CSC=C3) NC (=O) NC4=CC=CC (=C4) C (F) (F) F

Molecular Formula

C21 H18 F3 N3 O3 S2

Additionnal Information

AGI-6780 is a potent and selective inhibitor of IDH2 R140Q mutant with IC50 of 23 nM.

Storage Conditions

2 years -80 in solvent

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