Sulfaphenazole

Product Specifications

CAS Number

526-08-9

Synonyms

Depocid, Depotsulfonamide, Plisulfan, Raziosulfa

SKU

C17269-100mg

Target

P450 (e.g. CYP17)

Applications

Metabolism

Smiles

C1=CC=C (C=C1) N2C (=CC=N2) NS (=O) (=O) C3=CC=C (C=C3) N

Molecular Formula

C15H14N4O2S

Additionnal Information

Sulfaphenazole (Depocid, Depotsulfonamide, Plisulfan, Raziosulfa) is an inhibitor of CYP2C9 with Ki value of 0.3 μM and demonstrates at least 100-fold selectivity over other CYP450 isoforms (Ki values of 63 and 29 μM for CYP2C8 and CYP2C18, respectively, and no activity at CYP1A1, CYP1A2, CYP3A4, CYP2C19) .