Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Pelitinib (EKB-569)

Product Specifications

CAS Number

257933-82-7

SKU

C16291-100mg

Target

EGFR

Applications

Protein Tyrosine Kinase

Smiles

CCOC1=C (C=C2C (=C1) N=CC (=C2NC3=CC (=C (C=C3) F) Cl) C#N) NC (=O) C=CCN (C) C

Molecular Formula

C24H23ClFN5O2

Additionnal Information

Pelitinib (EKB-569) is a potent irreversible EGFR inhibitor with IC50 of 38.5 nM. Pelitinib (EKB-569) also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282 nM, 800 nM and 1255 nM, respectively. Phase2.

Storage Conditions

2 years -80 in solvent

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Epsin 2 (EPN2) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI1G3]
TA504296AM 100 µL

Epsin 2 (EPN2) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI1G3]

Sign In for Pricing
View Details
EXOSC9 Recombinant Rabbit Monoclonal Antibody [PSH08-55]
HA723001 100 µL

EXOSC9 Recombinant Rabbit Monoclonal Antibody [PSH08-55]

Sign In for Pricing
View Details
Human Angiotensinogen, C-His Tag
HA211165-01 20 µg

Human Angiotensinogen, C-His Tag

Sign In for Pricing
View Details
Human Angiotensinogen, C-His Tag
HA211165-02 50 µg

Human Angiotensinogen, C-His Tag

Sign In for Pricing
View Details
Human Angiotensinogen, C-His Tag
HA211165-03 100 µg

Human Angiotensinogen, C-His Tag

Sign In for Pricing
View Details
PPA2 (NM_001034191) Human Over-expression Lysate
LC421959 20 µg

PPA2 (NM_001034191) Human Over-expression Lysate

Sign In for Pricing
View Details