Elzovantinib (TPX-0022)
Product Specifications
CAS Number
2271119-26-5
Synonyms
CSF1R-IN-2
SKU
C14367-5mg
Target
C-Met
Applications
Protein Tyrosine Kinase
Molecular Formula
C20H20FN7O2
Additionnal Information
Elzovantinib (TPX-0022, CSF1R-IN-2) is a potent inhibitor of MET/CSF1R/SRC with enzymatic kinase inhibition IC50s of 0.14 nM, 0.71 nM and 0.12 nM, respectively. TPX-0022 modulates the tumor immune microenvironment in preclinical models.
Storage Conditions
3 years -20°C powder
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