What is the catalog number for ML221?

The catalog number for ML221 is C13597.

What sizes are available for ML221?

ML221 is available in the following size(s): 10 mg, 100 mg.

How many pack sizes does ML221 come in?

ML221 is available in 2 different pack sizes.

ML221 is currently made to order / not held in immediate stock. Contact us for lead time.

Are there any special shipping requirements for ML221?

ML221 is requires dry ice shipping.

ML221

Product Specifications

CAS Number

877636-42-5

SKU

C13597-10mg

Target

Angiotensin Receptor

Applications

GPCR & G Protein

Smiles

C1=CN=C (N=C1) SCC2=CC (=O) C (=CO2) OC (=O) C3=CC=C (C=C3) [N+] (=O) [O-]

Molecular Formula

C17H11N3O6S

Additionnal Information

ML221 is a potent apelin receptor (APJ) functional antagonist in cell-based assays that is >37-fold selective over the closely related angiotensin II type 1 (AT1) receptor. The IC50 values of ML221 are 0.70 and 1.75 μM in a cAMP assay and β-arrestin assay, respectively.