What is the catalog number for Tolinapant (ASTX660)?

The catalog number for Tolinapant (ASTX660) is C13586.

What sizes are available for Tolinapant (ASTX660)?

Tolinapant (ASTX660) is available in the following size(s): 1 mg, 5 mg, 10 mM / 1 mL, 100 mg.

How many pack sizes does Tolinapant (ASTX660) come in?

Tolinapant (ASTX660) is available in 4 different pack sizes.

Is Tolinapant (ASTX660) in stock?

Tolinapant (ASTX660) is currently made to order / not held in immediate stock. Contact us for lead time.

Tolinapant (ASTX660)

Product Specifications

CAS Number

1799328-86-1

SKU

C13586-1mg

Target

IAP

Applications

Apoptosis

Smiles

CC1CN (C (CN1) CN2CCOCC2C) CC (=O) N3CC (C4=C3C=C (C (=N4) CO) CC5=CC=C (C=C5) F) (C) C

Molecular Formula

C30H42FN5O3

Additionnal Information

Tolinapant (ASTX660) is a potent, non-peptidomimetic antagonist of cIAP1/2 and XIAP that inhibits the interactions between a SMAC-derived peptide and the BIR3 domains of XIAP (BIR3-XIAP) and cIAP1 (BIR3-cIAP1) with IC50 values less than 40 and 12 nmol/L, respectively.