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Pemrametostat (GSK3326595)

Product Specifications

CAS Number

1616392-22-3

Synonyms

EPZ015938

SKU

C13572-5mg

Target

Histone Methyltransferase

Applications

Epigenetics

Smiles

CC (=O) N1CCC (CC1) NC2=NC=NC (=C2) C (=O) NCC (CN3CCC4=CC=CC=C4C3) O

Molecular Formula

C24H32N6O3

Additionnal Information

Pemrametostat (GSK3326595, EPZ015938) is an orally active, potent and selective inhibitor of protein arginine methyltransferase 5 (PRMT5) and potently inhibits tumor growth in vitro and in vivo in animal models.

Storage Conditions

2 years -80 in solvent

Available Sizes

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