EED226
Product Specifications
CAS Number
2083627-02-3
SKU
C13450-5mg
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CS (=O) (=O) C1=CC=C (C=C1) C2=CN=C (N3C2=NN=C3) NCC4=CC=CO4
Molecular Formula
C17H15N5O3S
Additionnal Information
EED226 is a potent, selective, and orally bioavailable a novel allosteric Polycomb repressive complex 2 (PRC2) inhibitor with an IC50 of 23.4 nM when the H3K27me0 peptide was used as substrate and an IC50 of 53.5 nM when the mononucleosome was used as the substrate. It directly binds to the H3K27me3 binding pocket of EED.
Storage Conditions
2 years -80 in solvent
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
GTR15385792 1 Vial
Lentiviral human SLC39A14 sgRNA gene knockout kit - Lentiviral human SLC39A14 sgRNA gene knockout kit (100)
Sign In for Pricing
View Details 168708-ML750 100 µL
CD56 (NCAM1, NCAM, Leu-19, NKH1, MSK39, NCAM120, NCAM140, NCAM180, Neural Cell Adhesion Molecule) (MaxLight 750) discontinued
Sign In for Pricing
View Details 