AZD5153 6-hydroxy-2-naphthoic acid
Product Specifications
CAS Number
1869912-40-2
Synonyms
AZD5153 HNT salt
SKU
C13358-5mg
Target
Epigenetic Reader Domain
Applications
Epigenetics
Smiles
CC1C (=O) N (CCN1CCOC2=CC=C (C=C2) C3CCN (CC3) C4=NN5C (=NN=C5OC) C=C4) C.C1=CC2=C (C=CC (=C2) O) C=C1C (=O) O
Molecular Formula
C25H33N7O3.C11H8O3
Additionnal Information
AZD5153 6-hydroxy-2-naphthoic acid (HNT salt) is a potent, selective, and orally available BET/BRD4 bromodomain inhibitor with pKi of 8.3 for BRD4. AZD5153 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes. NSD3, via H3K36me2, acts as an epigenetic deregulator to facilitate the expression of oncogenesis-promoting genes.
Storage Conditions
2 years -80 in solvent
Available Sizes
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
![Mouse Monoclonal EpCAM/TROP1 Antibody (rVU-1D9) [Allophycocyanin]](https://cdn.genprice.uk/genprice/uk/genprice4.webp)
NBP2-54408APC 100 µL
Mouse Monoclonal EpCAM/TROP1 Antibody (rVU-1D9) [Allophycocyanin]
Ask
View Details 
MBS2080438-01 0.1 mL
APC/CY7-Linked Polyclonal Antibody to Interleukin 1 Receptor Like Protein 1 (IL1RL1)
Ask
View Details 
MBS2080438-02 0.2 mL
APC/CY7-Linked Polyclonal Antibody to Interleukin 1 Receptor Like Protein 1 (IL1RL1)
Ask
View Details MBS2080438-03 0.5 mL
APC/CY7-Linked Polyclonal Antibody to Interleukin 1 Receptor Like Protein 1 (IL1RL1)
Ask
View Details MBS2080438-04 1 mL
APC/CY7-Linked Polyclonal Antibody to Interleukin 1 Receptor Like Protein 1 (IL1RL1)
Ask
View Details MBS2080438-05 5 mL
APC/CY7-Linked Polyclonal Antibody to Interleukin 1 Receptor Like Protein 1 (IL1RL1)
Ask
View Details