Paxalisib (GDC-0084)

Product Specifications

CAS Number

1382979-44-3

Synonyms

RG7666

SKU

C13229-5mg

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

CC1 (C2=NC3=C (N2CCO1) N=C (N=C3N4CCOCC4) C5=CN=C (N=C5) N) C

Molecular Formula

C18H22N8O2

Additionnal Information

Paxalisib (GDC-0084, RG7666) is a brain penetrant inhibitor of PI3K and mTOR with Kiapp values of 2 nM, 46 nM, 3 nM, 10 nM and 70 nM for PI3Kα, PI3Kβ, PI3Kδ, PI3Kγ and mTOR.

Storage Conditions

2 years -80 in solvent

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

TL512431V 500 µL Each

Allc Mouse shRNA Lentiviral Particle (Locus ID 94041)

Ask

View Details

458557-01 100 mg

N-Cyclohexyl-4-bromo-3-methylbenzamide

Ask

View Details

458557-02 250 mg

N-Cyclohexyl-4-bromo-3-methylbenzamide

Ask

View Details

NB100-53810 0.1 mg

Goat Polyclonal Cytochrome P450 26B1 Antibody

Ask

View Details

TA381163 100 µL

RRP36 Rabbit Polyclonal Antibody

Ask

View Details

AM06343SU-N 100 µL

MPS1 (RPS27) Mouse Monoclonal Antibody [Clone ID: 7E3]

Ask

View Details