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AZD8835

Product Specifications

CAS Number

1620576-64-8

SKU

C13090-5mg

Target

PI3K

Applications

PI3K/Akt/mTOR

Smiles

CCN1C (=NC (=N1) C2CCN (CC2) C (=O) CCO) C3=CN=C (C (=N3) C4=NN=C (O4) C (C) (C) C) N

Molecular Formula

C22H31N9O3

Additionnal Information

AZD8835 ia a novel mixed inhibitor of PI3Kα and PI3Kδ with IC50 of 6.2 nM and 5.7 nM, respectively, also with selectivity against PI3Kβ (IC50=431 nM) and PI3Kγ (IC50=90 nM) .

Storage Conditions

2 years -80 in solvent

Available Sizes

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