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Epacadostat (INCB024360)

Product Specifications

CAS Number

1204669-58-8

SKU

C13043-5mg

Target

IDO/TDO

Applications

Metabolism

Smiles

C1=CC (=C (C=C1N=C (C2=NON=C2NCCNS (=O) (=O) N) NO) Br) F

Molecular Formula

C11H13BrFN7O4S

Additionnal Information

Epacadostat (INCB024360) is a potent and selective indoleamine 2,3-dioxygenase (IDO1) inhibitor with IC50 of 10 nM and displays high selectivity over other related enzymes such as IDO2 or tryptophan 2,3-dioxygenase (TDO) .

Storage Conditions

2 years -80 in solvent

Available Sizes

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