Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Pelabresib (CPI-0610)

Product Specifications

CAS Number

1380087-89-7

SKU

C13001-5mg

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CC1=NOC2=C1C3=CC=CC=C3C (=NC2CC (=O) N) C4=CC=C (C=C4) Cl

Molecular Formula

C20H16ClN3O2

Additionnal Information

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.

Storage Conditions

2 years -80 in solvent

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

SOX10 (SOX10/1074), CF647 conjugate, 0.1mg/mL
BNC471017-500 1x 500 µL

SOX10 (SOX10/1074), CF647 conjugate, 0.1mg/mL

Sign In for Pricing
View Details
3Beta-Hydroxyandrosta-5,15-dien-17-one
TRC-H750020-10MG 10 mg

3Beta-Hydroxyandrosta-5,15-dien-17-one

Sign In for Pricing
View Details
EOLA1 (NM_001171909) Human Over-expression Lysate
LY432583 100 µg

EOLA1 (NM_001171909) Human Over-expression Lysate

Sign In for Pricing
View Details
ASB6 (NM_017873) Human Recombinant Protein
TP309519L 1 mg

ASB6 (NM_017873) Human Recombinant Protein

Sign In for Pricing
View Details
Ferritin, Light Chain (FTL) (Microglia Marker) (FTL/2338R), CF568 conjugate, 0.1mg/mL
BNC682338-500 1x 500 µL

Ferritin, Light Chain (FTL) (Microglia Marker) (FTL/2338R), CF568 conjugate, 0.1mg/mL

Sign In for Pricing
View Details
Tissue FFPE Sections, Ovary: right
CS700339 5x 5 µm

Tissue FFPE Sections, Ovary: right

Sign In for Pricing
View Details