Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

Pelabresib (CPI-0610)

Product Specifications

CAS Number

1380087-89-7

SKU

C13001-5mg

Target

Epigenetic Reader Domain

Applications

Epigenetics

Smiles

CC1=NOC2=C1C3=CC=CC=C3C (=NC2CC (=O) N) C4=CC=C (C=C4) Cl

Molecular Formula

C20H16ClN3O2

Additionnal Information

Pelabresib (CPI-0610) is a potent and selective benzoisoxazoloazepine BET bromodomain inhibitor with an IC50 of 39 nM for BRD4-BD1 in TR-FRET assay and currently undergoing human clinical trials for hematological malignancies. CPI-0610 inhibits the expression of Nuclear receptor binding SET domain protein 3 (NSD3) target genes.

Storage Conditions

2 years -80 in solvent

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Tissue FFPE Sections, Lung
CS802127 5x 5 µm

Tissue FFPE Sections, Lung

Sign In for Pricing
View Details
Glutaminase (GLS) (NM_014905) Human Recombinant Protein
TP306265M 100 µg

Glutaminase (GLS) (NM_014905) Human Recombinant Protein

Sign In for Pricing
View Details
Perfluorohexanes (Mixture of Isomers)
TRC-P999223-1G 1 g

Perfluorohexanes (Mixture of Isomers)

Sign In for Pricing
View Details
Cytokeratin, LMW (AE-1), CF740 conjugate, 0.1mg/mL
BNC740253-500 1x 500 µL

Cytokeratin, LMW (AE-1), CF740 conjugate, 0.1mg/mL

Sign In for Pricing
View Details
Purified Rat IgG2b, κ Isotype Control[LTF-2]
E-AB-F09843A-01 25 µg

Purified Rat IgG2b, κ Isotype Control[LTF-2]

Sign In for Pricing
View Details
Purified Rat IgG2b, κ Isotype Control[LTF-2]
E-AB-F09843A-02 100 µg

Purified Rat IgG2b, κ Isotype Control[LTF-2]

Sign In for Pricing
View Details